19 patents
Utility
Quinazolines, Pharmaceutical Compositions, and Therapeutic Applications
21 Sep 23
Paul E. Erdman, Leah M. Fung, Patrick Papa, Brandon Whitefield
Filed: 15 Mar 23
Utility
PDE4 Inhibitors, Pharmaceutical Compositions, and Therapeutic Applications
9 Mar 23
Kyle W.H. Chan, Paul E. Erdman, Leah M. Fung, David Aaron Hecht, Frank Mercurio, Robert W. Sullivan
Filed: 14 Dec 20
Utility
Pyrazolylpyrimidines and Use Thereof
16 Feb 23
Kyle W.H. Chan, Robert W. Sullivan
Filed: 12 Jan 21
Utility
Ras Protein Degraders, Pharmaceutical Compositions Thereof, and Their Therapeutic Applications
5 Jan 23
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah M. Fung, David Aaron Hecht, Imelda Lam, Frank Mercurio, Robert W. Sullivan, Eduardo Torres
Filed: 14 Sep 20
Utility
Protein-targeting Compounds and Pharmaceutical Compositions Thereof, and Their Therapeutic Applications
22 Sep 22
Kyle W.H. Chan, Paul E. Erdman, Aparajita Hoskote Chourasia, Leah M. Fung, David Aaron Hecht, Imelda Lam, Frank Mercurio, Robert W. Sullivan, Eduardo Torres
Filed: 30 May 22
Utility
Fused Thiophene Compounds
24 Mar 22
The present disclosure provides compounds that modulate protein function, to restore protein homeostasis, and cell-cell adhesion.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah M. Fung, Frank Mercurio, Robert W. Sullivan
Filed: 6 Dec 21
Utility
Aminoamide Compounds
20 May 21
Compounds with amino amide linkers and pharmaceutical compositions and medicaments comprising such compounds are disclosed.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah M. Fung, Frank Mercurio, Robert W. Sullivan
Filed: 1 Feb 21
Utility
Compounds Targeting Proteins, Compositions, Methods, and Uses Thereof
13 May 21
The present invention provides compounds that modulate protein function, to restore protein homeostasis, including cytokine, CKα, GSPT1, aiolos, and/or ikaros activity, and cell-cell adhesion.
Kyle W.H. Chan, Paul E. Erdman, Leah M. Fung, Frank Mercurio, Robert W. Sullivan, Eduardo Torres
Filed: 11 Jan 21
Utility
Protein-targeting Compounds and Pharmaceutical Compositions Thereof, and Their Therapeutic Applications
25 Nov 20
Kyle W.H. Chan, Paul E. Erdman, Aparajita Hoskote Chourasia, Leah Fung, David Aaron Hecht, Imelda Lam, Frank Mercurio, Robert Sullivan, Eduardo Torres
Filed: 25 May 20
Utility
Substituted Isoindolinones
14 Oct 20
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah M. Fung, Imelda Lam, Frank Mercurio, Robert W. Sullivan, Eduardo Torres
Filed: 24 Jun 20
Utility
Ether Compounds and Uses Thereof
22 Jul 20
The present invention provides compounds that modulate protein function, to restore protein homeostasis and/or cell-cell adhesion.
Kyle W.H. Chan, Frank Mercurio, Aparajita Hoskote Chourasia, Leah Fung, Robert Sullivan
Filed: 17 Dec 19
Utility
Bicyclic Compounds and Methods of Use
3 Jun 20
The present invention provides compounds that modulate protein function, specifically phosphodiesterase 4 (PDE4).
Robert Sullivan, Paul E. Erdman, Eduardo Torres, Leah Fung, Kyle W.H. Chan, Frank Mercurio
Filed: 10 Feb 20
Utility
Substituted Isoindolinones
13 May 20
Substituted isoindolinones of Formula (I), methods of making such compounds, pharmaceutical compositions and medicaments comprising such compounds, and methods of using such compounds to treat or ameliorate diseases, disorders, or conditions associated with protein malfunction, such as cancer, are provided.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah Fung, Imelda Lam, Frank Mercurio, Robert Sullivan, Eduardo Torres
Filed: 11 Nov 19
Utility
Bifunctional Compounds
12 Feb 20
The present application provides compounds that modulate CDK protein function.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah Fung, David Aaron Hecht, Frank Mercurio, Robert Sullivan, Joseph P. Vacca
Filed: 24 Jul 19
Utility
Aminoamide Compounds
8 Jan 20
Compounds with amino amide linkers and pharmaceutical compositions and medicaments comprising such compounds are disclosed.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah Fung, Frank Mercurio, Robert Sullivan
Filed: 10 Jun 19
Utility
Fused Thiophene Compounds
1 Jan 20
The present disclosure provides compounds that modulate protein function, to restore protein homeostasis, and cell-cell adhesion.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah Fung, Frank Mercurio, Robert Sullivan
Filed: 10 Jun 19
Utility
Compounds Targeting Proteins, Compositions, Methods, and Uses Thereof
4 Dec 19
The present invention provides modulators of protein function, to restore protein homeostasis, including GSPT1 activity.
Kyle W.H. Chan, Paul E. Erdman, Leah Fung, Frank Mercurio, Robert Sullivan
Filed: 12 Aug 19
Utility
Compounds Targeting Proteins, Compositions, Methods, and Uses Thereof
23 Oct 19
The present invention provides compounds that modulate protein function, to restore protein homeostasis, including cytokine, CK1α, GSPT1, aiolos, and/or ikaros activity, and cell-cell adhesion.
Kyle W.H. Chan, Paul E. Erdman, Leah Fung, Frank Mercurio, Robert Sullivan, Eduardo Torres
Filed: 27 Jun 19
Utility
Thienopyrimidinone Compounds
23 Oct 19
The present disclosure provides compounds that modulate protein function and/or restore protein homeostasis.
Kyle W.H. Chan, Aparajita Hoskote Chourasia, Paul E. Erdman, Leah Fung, Imelda Lam, Frank Mercurio, Robert Sullivan, Eduardo Torres
Filed: 27 Mar 19
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